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Found 3 results for OCT1 HEK293.
Service
Transporters
...solubility assessment at an additional charge. Percent inhibition is calculated as 100 x [1-(IROCT1-IRVC)TC / (IROCT1 – IRVC)0], where IROCT1 is the influx rate of MPP+ in OCT1-transfected cells, IRVC is the influx rate...
Service
Discovery in vitro ADMET
...OATP1B3, OAT1, OAT3, OCT1, OCT2, OATP2B1, OATP1A2, MATE1, MATE2, PEPT1, NTCP, ASBT) Hepatic uptake using media-loss method Download our poster about our permeability assay platform Metabolic Stability and Identification Metabolic...
Service
Regulatory in vitro ADMET Studies
...(PAMPA, Caco-2, MDCK and transfected MDCK cell lines) Transporter investigation on substrate and inhibitor evaluation (P-gp, BCRP, BSEP, MRP2, MRP3, MRP4, OATP1B1, OATP1B3, OTAP2B1, OAT1, OAT3, OCT1, OCT2, MATE1, MATE2K,...