Found 3 results for OAT3 HEK293.

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Transporters

...OAT3 probe substrate PAH at 10 μM Test compound at six concentrations (serial diluations from 100 µM) in modified Hanks’ buffer with less than 0.8% DMSO Assay System OAT3-transfected HEK293...
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Regulatory in vitro ADMET Studies

...(PAMPA, Caco-2, MDCK and transfected MDCK cell lines) Transporter investigation on substrate and inhibitor evaluation (P-gp, BCRP, BSEP, MRP2, MRP3, MRP4, OATP1B1, OATP1B3, OTAP2B1, OAT1, OAT3, OCT1, OCT2, MATE1, MATE2K,...
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Discovery in vitro ADMET

...OATP1B1, OATP1B3, OAT1, OAT3, OCT1, OCT2, OATP2B1, OATP1A2, MATE1, MATE2, PEPT1, NTCP, ASBT) Hepatic uptake using media-loss method Download our poster about our permeability assay platform Metabolic Stability and Identification...